Distribution of amantadine-resistant H5N1 avian influenza variants in Asia.

Cheung, Chung-Lam; Rayner, Jane M; Smith, Gavin J D; Wang, Pui; Naipospos, T S P; Zhang, Jinxia; Yuen, Kwok-Yung; Webster, Robert G et al. · J Infect Dis · 2006

basic_science · Level V

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Abstract

We examined the distribution of genetic mutations associated with resistance to the M2 ion channel-blocking adamantane derivatives, amantadine and rimantadine, among H5N1 viruses isolated in Vietnam, Thailand, Cambodia, Indonesia, Hong Kong, and China. More than 95% of the viruses isolated in Vietnam and Thailand contained resistance mutations, but resistant mutants were less commonly isolated in Indonesia (6.3% of isolates) and China (8.9% of isolates), where human infection was recently reported. The dual mutation motif Leu26Ile-Ser31Asn (leucine-->isoleucine at aa 26 and serine-->asparagine at aa 31) was found almost exclusively in all resistant isolates from Vietnam, Thailand, and Cambodia, suggesting the biological selection of these mutations.

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