MSN-mediated sequential vascular-to-cell nuclear-targeted drug delivery for efficient tumor regression.

Pan, Limin; Liu, Jianan; He, Qianjun; Shi, Jianlin · Adv Mater · 2014

basic_science · Level V

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Abstract

Mesoporous silica nanoparticles functionalized with peptides are developed for sequential drug delivery. The RGD peptide is used for vasculature/cell membrane targeting and the TAT peptide for nuclear targeting. Using this delivery strategy, a tumor in a murine xenograft model is successfully regressed.

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