BAD and K<sub>ATP</sub> channels regulate neuron excitability and epileptiform activity.

Martínez-François, Juan Ramón; Fernández-Agüera, María Carmen; Nathwani, Nidhi; Lahmann, Carolina; Burnham, Veronica L; Danial, Nika N; Yellen, Gary · Elife · 2018

basic_science · Level V

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Abstract

Brain metabolism can profoundly influence neuronal excitability. Mice with genetic deletion or alteration of <i>Bad</i> (<u>B</u>CL-2 <u>a</u>gonist of cell <u>d</u>eath) exhibit altered brain-cell fuel metabolism, accompanied by resistance to acutely induced epileptic seizures; this seizure protection is mediated by ATP-sensitive potassium (K<sub>ATP</sub>) channels. Here we investigated the effect of BAD manipulation on K<sub>ATP</sub> channel activity and excitability in acute brain slices. We found that BAD's influence on neuronal K<sub>ATP</sub> channels was cell-autonomous and directly affected dentate granule neuron (DGN) excitability. To investigate the role of neuronal K<sub>ATP</sub> channels in the anticonvulsant effects of BAD, we imaged calcium during picrotoxin-induced epileptiform activity in entorhinal-hippocampal slices. BAD knockout reduced epileptiform activity, and this effect was lost upon knockout or pharmacological inhibition of K<sub>ATP</sub> channels. Targeted BAD knockout in DGNs alone was sufficient for the antiseizure effect in slices, consistent with a 'dentate gate' function that is reinforced by increased K<sub>ATP</sub> channel activity.

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