Goldilocks Dosing of TKIs: A Dose that Is Just Right Leads to Optimal Outcomes.

Rini, Brian I · Clin Cancer Res · 2018

editorial · Level V

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Abstract

Higher concentrations of TKIs, such as pazopanib, are associated with improved outcomes in advanced RCC. A phase III trial failed to show disease-free survival benefit to pazopanib in the adjuvant setting, but improved DFS was seen in patients with higher <i>C</i><sub>trough</sub> levels, supporting adequate drug exposure for optimal clinical outcome. <i>Clin Cancer Res; 24(13); 2979-80. ©2018 AACR</i><i>See related article by Sternberg et al., p. 3005</i>.

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