Suppression of angiopoietin-like 4 reprograms endothelial cell metabolism and inhibits angiogenesis.

Chaube, Balkrishna; Citrin, Kathryn M; Sahraei, Mahnaz; Singh, Abhishek K; de Urturi, Diego Saenz; Ding, Wen; Pierce, Richard W; Raaisa, Raaisa et al. · Nat Commun · 2023

basic_science · Level V

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Abstract

Angiopoietin-like 4 (ANGPTL4) is known to regulate various cellular and systemic functions. However, its cell-specific role in endothelial cells (ECs) function and metabolic homeostasis remains to be elucidated. Here, using endothelial-specific Angptl4 knock-out mice (Angptl4<sup>iΔEC</sup>), and transcriptomics and metabolic flux analysis, we demonstrate that ANGPTL4 is required for maintaining EC metabolic function vital for vascular permeability and angiogenesis. Knockdown of ANGPTL4 in ECs promotes lipase-mediated lipoprotein lipolysis, which results in increased fatty acid (FA) uptake and oxidation. This is also paralleled by a decrease in proper glucose utilization for angiogenic activation of ECs. Mice with endothelial-specific deletion of Angptl4 showed decreased pathological neovascularization with stable vessel structures characterized by increased pericyte coverage and reduced permeability. Together, our study denotes the role of endothelial-ANGPTL4 in regulating cellular metabolism and angiogenic functions of EC.

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